1   2   3   4   5   6   7   8   9   10   11   12  
Design, synthesis and biological evaluation of novel 2,4-thiazolidinedione derivatives able to target the human BAG3 protein
Budassi, Federica; Marchioro, Chiara; Canton, Martina; Favaro, Annagiulia; Sturlese, Mattia; Urbinati, Chiara; Rusnati, Marco; Romagnoli, Romeo; Viola, Giampietro; Mariotto, Elena     details >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 261, No. 1, pp: 115824-115824, Anno: 2023

Development of a clot-adhesive coating to improve the performance of thrombectomy devices
Skarbek, Charles; Anagnostakou, Vania; Procopio, Emanuele; Epshtein, Mark; Raskett, Christopher M; Romagnoli, Romeo; Iviglia, Giorgio; Morra, Marco; Antonucci, Marta; Nicoletti, Antonino; Caligiuri, Giuseppina; Gounis, Matthew J     details >>
JOURNAL OF NEUROINTERVENTIONAL SURGERY
Vol. 15, No. 12, pp: 1207-1211, Anno: 2023

Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a sulfanilamide scaffold
Romagnoli, Romeo; De Ventura, Tiziano; Manfredini, Stefano; Baldini, Erika; Supuran, Claudiu T; Nocentini, Alessio; Brancale, Andrea; Bortolozzi, Roberta; Manfreda, Lorenzo; Viola, Giampietro     details >>
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Vol. 38, No. 1, pp: 2270180-2270180, Anno: 2023

Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents
Oliva, Paola; Romagnoli, Romeo; Cacciari, Barbara; Manfredini, Stefano; Padroni, Chiara; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Milan, Noemi; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta     details >>
PHARMACEUTICS
Vol. 14, No. 6, pp: 1191-1-1191-44, Anno: 2022

Cinnamic acid derivatives linked to arylpiperazines as novel potent inhibitors of tyrosinase activity and melanin synthesis
Romagnoli, Romeo; Oliva, Paola; Prencipe, Filippo; Manfredini, Stefano; Germanò, Maria Paola; De Luca, Laura; Ricci, Federico; Corallo, Diana; Aveic, Sanja; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta     details >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 231, No. 1, pp: 114147-1-114147-16, Anno: 2022

Design, Synthesis and Biological Investigation of 2-Anilino Triazolopyrimidines as Tubulin Polymerization Inhibitors with Anticancer Activities
Romagnoli, Romeo; Oliva, Paola; Prencipe, Filippo; Manfredini, Stefano; Budassi, Federica; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Manfreda, Lorenzo; Mariotto, Elena; Bortolozzi, Roberta; Viola, Giampietro     details >>
PHARMACEUTICALS
Vol. 15, No. 8, pp: 1031-1-1031-29, Anno: 2022

Synergistic Effects of A Combined Treatment of Glioblastoma U251 Cells with An Anti-miR-10b-5p Molecule and An AntiCancer Agent Based on 1-(3',4',5'-Trimethoxyphenyl)-2-Aryl-1H-Imidazole Scaffold
Zurlo, Matteo; Romagnoli, Romeo; Oliva, Paola; Gasparello, Jessica; Finotti, Alessia; Gambari, Roberto     details >>
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
Vol. 23, No. 11, pp: 5991-1-5991-15, Anno: 2022

Thio-substituted derivatives of 4-amino-pyrazolo[3,4-d]pyrimidine-6-thiol as antiproliferative agents
Cacciari, B.; Romagnoli, R.; Romani, A.; Trentini, A.; Hanau, S.     details >>
FUTURE MEDICINAL CHEMISTRY
Vol. 13, No. 18, pp: 1515-1530, Anno: 2021

A Facile Synthesis of Diaryl Pyrroles Led to the Discovery of Potent Colchicine Site Antimitotic Agents
Romagnoli, Romeo; Oliva, Paola; Salvador, Maria Kimatrai; Manfredini, Stefano; Padroni, Chiara; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Maccarinelli, Federica; Rruga, Fatlum; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta     details >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 214, No. 1, pp: 113229-1-113229-20, Anno: 2021

Apoptosis Pathways Triggered by a Potent Antiproliferative Hybrid Chalcone on Human Melanoma Cells
Rodríguez, Irene; Saavedra, Ester; del Rosario, Henoc; Perdomo, Juan; Quintana, José; Prencipe, Filippo; Oliva, Paola; Romagnoli, Romeo; Estévez, Francisco     details >>
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
Vol. 22, No. 24, pp: 13462-1-13462-19, Anno: 2021

Synergistic effects of the combined treatment of U251 and T98G glioma cells with an anti-tubulin tetrahydrothieno[2,3-c]pyridine derivative and a peptide nucleic acid targeting miR-221-3p
Zurlo, M.; Romagnoli, R.; Oliva, P.; Gasparello, J.; Finotti, A.; Gambari, R.     details >>
INTERNATIONAL JOURNAL OF ONCOLOGY
Vol. 59, No. 2, pp: 61-1-61-13, Anno: 2021

Concise synthesis and biological evaluation of 2-Aryl-3-Anilinobenzo[b]thiophene derivatives as potent apoptosis-inducing agents
Romagnoli, Romeo; Preti, Delia; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro; Brancale, Andrea; Ferla, Salvatore; Morciano, Giampaolo; Pinton, Paolo     details >>
BIOORGANIC CHEMISTRY
Vol. 112, No. 1, pp: 104919-1-104919-15, Anno: 2021

Synthesis and biological evaluation of new antitubulin agents containing 2-(30,40,50-trimethoxyanilino)-3,6-disubstituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine Scaffold
Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Cacciari, Barbara; Balzarini, Jan; Liekens, Sandra; Hamel, Ernest; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Zurlo, Matteo; Finotti, Alessia; Gambari, Roberto     details >>
MOLECULES
Vol. 25, No. 7, pp: 1690-1-1690-23, Anno: 2020

Synthesis and biological evaluation of 2-substituted benzyl-/phenylethylamino-4-amino-5-aroylthiazoles as apoptosis-inducing anticancer agents
Oliva, Paola; Onnis, Valentina; Balboni, Elisa; Hamel, Ernest; Estévez-Sarmiento, Francisco; Quintana, José; Estévez, Francisco; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Romagnoli, Romeo     details >>
MOLECULES
Vol. 25, No. 9, pp: 2177-1-2177-18, Anno: 2020

Thioridazine requires calcium influx to induce MLL-AF6-rearranged AML cell death
Tregnago, Claudia; Da Ros, Ambra; Porcù, Elena; Benetton, Maddalena; Simonato, Manuela; Simula, Luca; Borella, Giulia; Polato, Katia; Minuzzo, Sonia; Borile, Giulia; Cogo, Paola; Campello, Silvia; Massi, Alessandro; Romagnoli, Romeo; Buldini, Barbara; Locatelli, Franco; Pigazzi, Martina     details >>
BLOOD ADVANCES
Vol. 4, No. 18, pp: 4417-4429, Anno: 2020

The Detrimental Action of Adenosine on Glutamate-Induced Cytotoxicity in PC12 Cells Can Be Shifted towards a Neuroprotective Role through A1AR Positive Allosteric Modulation
Vincenzi, F.; Pasquini, S.; Gessi, S.; Merighi, S.; Romagnoli, R.; Borea, P. A.; Varani, K.     details >>
CELLS
Vol. 9, No. 5, pp: 1242-1-1242-16, Anno: 2020

Design, synthesis and biological evaluation of 2-alkoxycarbonyl-3-anilinoindoles as a new class of potent inhibitors of tubulin polymerization
Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Kimatrai Salvador, Maria; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Viola, Giampietro; Bortolozzi, Roberta; Persoons, Leentje; Balzarini, Jan; Liekens, Sandra; Schols, Dominique     details >>
BIOORGANIC CHEMISTRY
Vol. 97, No. April 2020, pp: 103665-1-103665-18, Anno: 2020

Design, synthesis, in vitro and in vivo biological evaluation of 2-amino-3-aroylbenzo[b]furan derivatives as highly potent tubulin polymerization inhibitors
Oliva, Paola; Romagnoli, Romeo; Manfredini, Stefano; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Maccarinelli, Federica; Giacomini, Arianna; Rruga, Fatlum; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta     details >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 200, No. 15 August 2020, pp: 112448-1-112448-17, Anno: 2020

Design, Synthesis, and Biological Evaluation of 6-Substituted Thieno[3,2-d]pyrimidine Analogues as Dual Epidermal Growth Factor Receptor Kinase and Microtubule Inhibitors
Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Schiaffino Ortega, Santiago; Chayah, Mariem; Kimatrai Salvador, Maria; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Mattiuzzo, Elena; Viola, Giampietro     details >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 62, No. 3, pp: 1274-1290, Anno: 2019

Design, synthesis and biological evaluation of novel vicinal diaryl-substituted 1H-Pyrazole analogues of combretastatin A-4 as highly potent tubulin polymerization inhibitors
Romagnoli, Romeo; Oliva, Paola; Salvador, Maria Kimatrai; Camacho, Maria Encarnacion; Padroni, Chiara; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Grillo, Elisabetta; Bortolozzi, Roberta; Rruga, Fatlum; Mariotto, Elena; Viola, Giampietro     details >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 181, No. 1, pp: 11577-1-11577-21, Anno: 2019

1   2   3   4   5   6   7   8   9   10   11   12